<p>Β-glucosidase, a ubiquitous enzyme, is responsible for catalyzing the hydrolysis of β-glycosidic linkages present in polysaccharides and contributes significantly to several industrial sectors such as food, agriculture, and biofuel production. β-glucosidases can convert polydatin to resveratrol through de-glycosylation. Resveratrol is important for human health and has potential applications in pharmacology. The preference of enzymatic conversion methods for resveratrol production improves the importance of β-glucosidases. The glucose tolerance of β-glucosidases also significantly impacts their applicability. Because the inhibition of many β-glucosidase’s activity by their reaction product, glucose, is a limiting factor for industrial applications. In this study, a robust β-glucosidase was isolated from a novel-defined <i>Jiangella ureilytica</i> KC603 strain. The β-glucosidase encoding gene (<i>JurBglKC603</i>) was cloned and expressed in <i>E. coli</i> BL21 (DE3) cells and a 50.1&#xa0;kDa protein was purified using Ni-affinity column chromatography. The efficient polydatin deglycosylation capacity of JurBglKC603 was determined by Glucose Oxidase–Peroxidase (GOPOD) assay. JurBglKC603 exhibits remarkable resistance to glucose concentrations of up to 3&#xa0;M. The enzyme remained active across a broad pH spectrum and was unaffected by most heavy metal ions, except for Hg<sup>2+</sup>. The kinetic parameters of JurBglKC603 were <i>K</i><sub>m</sub> = 0.44&#xa0;mM, <i>V</i><sub>max</sub> = 26.87 U·mg<sup>−1</sup>, <i>k</i><sub>cat</sub> = 21.1&#xa0;s<sup>−1</sup>, and <i>k</i><sub>cat</sub>/<i>K</i><sub>m</sub> = 47,954&#xa0;M<sup>−1</sup>·s<sup>−1</sup> against <i>p</i>NPG and <i>K</i><sub>m</sub> = 4.6&#xa0;mM, <i>V</i><sub>max</sub> = 20 U·mg<sup>−1</sup>, <i>k</i><sub>cat</sub> = 17.2&#xa0;s<sup>−1</sup>, and <i>k</i><sub>cat</sub>/<i>K</i><sub>m</sub> = 3822&#xa0;M<sup>−1</sup>·s<sup>−1</sup> against polydatin. Molecular docking studies have demonstrated that Gln19, His120, Trp411, and Glu410 play a vital role in the interaction with polydatin.</p>

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Biochemical Characterization of a Novel, Glucose-Tolerant β-Glucosidase from Jiangella ureilytica KC603, and Determination of Resveratrol Production Capacity from Polydatin

  • Arife Kaçıran,
  • Miray Şahinkaya,
  • Dilşat Nigar Çolak,
  • Numan Saleh Zada,
  • Murat Kaçağan,
  • Halil İbrahim Güler,
  • Hayrettin Saygın,
  • Ali Osman Beldüz

摘要

Β-glucosidase, a ubiquitous enzyme, is responsible for catalyzing the hydrolysis of β-glycosidic linkages present in polysaccharides and contributes significantly to several industrial sectors such as food, agriculture, and biofuel production. β-glucosidases can convert polydatin to resveratrol through de-glycosylation. Resveratrol is important for human health and has potential applications in pharmacology. The preference of enzymatic conversion methods for resveratrol production improves the importance of β-glucosidases. The glucose tolerance of β-glucosidases also significantly impacts their applicability. Because the inhibition of many β-glucosidase’s activity by their reaction product, glucose, is a limiting factor for industrial applications. In this study, a robust β-glucosidase was isolated from a novel-defined Jiangella ureilytica KC603 strain. The β-glucosidase encoding gene (JurBglKC603) was cloned and expressed in E. coli BL21 (DE3) cells and a 50.1 kDa protein was purified using Ni-affinity column chromatography. The efficient polydatin deglycosylation capacity of JurBglKC603 was determined by Glucose Oxidase–Peroxidase (GOPOD) assay. JurBglKC603 exhibits remarkable resistance to glucose concentrations of up to 3 M. The enzyme remained active across a broad pH spectrum and was unaffected by most heavy metal ions, except for Hg2+. The kinetic parameters of JurBglKC603 were Km = 0.44 mM, Vmax = 26.87 U·mg−1, kcat = 21.1 s−1, and kcat/Km = 47,954 M−1·s−1 against pNPG and Km = 4.6 mM, Vmax = 20 U·mg−1, kcat = 17.2 s−1, and kcat/Km = 3822 M−1·s−1 against polydatin. Molecular docking studies have demonstrated that Gln19, His120, Trp411, and Glu410 play a vital role in the interaction with polydatin.